SCHEMBL2904919

SCHEMBL2904919

COc1ccccc1C=CC(=O)N1CCC(=O)N(CCN2CCCC2)CC1

nearest known ligand 0.65

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.65
KDM4E B2RXH2 3/20 0.58
NFE2L2 Q16236 7/20 0.50
KEAP1 Q14145 5/20 0.50
NPC1 O15118 1/20 0.50
MAPT P10636 1/20 0.50
RAB9A P51151 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
ALDH1A1 P00352 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.47
TFEB P19484 1/20 0.46
PKM P14618 1/20 0.45
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
HTR2B P41595 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2904918 1.00 HPGD (0.65) HPGDKDM4ENFE2L2KEAP1NPC1
SCHEMBL2904853 0.82 MEN1 (0.58) HPGDKDM4ENPC1MAPTRAB9A
SCHEMBL2904849 0.82 MEN1 (0.58) HPGDKDM4ENPC1MAPTRAB9A
SCHEMBL2896752 0.82 GPR183 (0.56) NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL2896756 0.82 GPR183 (0.56) NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL3112646 0.79 HPGD (0.97) HPGDKDM4ENFE2L2NPC1MAPT
SCHEMBL3112643 0.79 HPGD (0.97) HPGDKDM4ENFE2L2NPC1MAPT
SCHEMBL2905043 0.79 APP (0.47) RAB9AALDH1A1
SCHEMBL2905040 0.79 APP (0.47) RAB9AALDH1A1
SCHEMBL2902873 0.78 ALDH1A1 (0.60) NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010506-B1 DIAZEPAN DERIVATIVES MODULATORS OF CHEMOKINE RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-04 EP disclosed