SCHEMBL29050355

SCHEMBL29050355

COc1ccc2ncc(Cl)c(C(=O)N3CCC3)c2n1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPGD P15428 6/20 0.47
LRRK2 Q5S007 5/20 0.41
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
NPC1 O15118 1/20 0.40
GLA P06280 1/20 0.40
PTK2 Q05397 1/20 0.39
GPR183 P32249 1/20 0.39
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38
HRH3 Q9Y5N1 1/20 0.37
CYP8B1 Q9UNU6 1/20 0.37
HTT P42858 1/20 0.36
TP53 P04637 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31391928 1.00 HPGD (0.47) HPGDLRRK2HCRTR1HCRTR2NPC1
SCHEMBL29050335 0.82 HPGD (0.37) HPGDGLAKCNH2
SCHEMBL29050321 0.82 POLB (0.42) KCNH2
SCHEMBL2038295 0.81 NNMT (0.44) KCNH2
SCHEMBL3155020 0.78 SMN1; SMN2 (0.37) KCNH2
SCHEMBL2766836 0.77 KCNH2 (0.35) HPGDNPC1HTTKCNH2
SCHEMBL30354542 0.73 DYRK1A (0.43) HPGDTP53KCNH2
SCHEMBL1075375 0.73 DYRK1A (0.36) HPGDNPC1HTTTP53KCNH2
SCHEMBL2770307 0.73 KCNH2 (0.36) KCNH2
SCHEMBL29692824 0.73 KCNH2 (0.36) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116528857-A MALT-1 modulators 艾克斯赛安西娅人工智能有限公司 2023-08-01 CN disclosed