SCHEMBL2905249

SCHEMBL2905249

Nc1nc2cccc(N)c2cc1C[C@H]1CCc2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.47
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
GLA P06280 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
PTBP1 P26599 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
RCE1 Q9Y256 1/20 0.40
ESR1 P03372 3/20 0.37
ESR2 Q92731 3/20 0.37
SLC22A1 O15245 1/20 0.34
PRCP P42785 1/20 0.34
TLR8 Q9NR97 4/20 0.34
APP P05067 1/20 0.34
MTNR1A P48039 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2242767 0.78 KDM4E (0.44) HTR6KDM4ENPC1ALDH1A1LMNA
SCHEMBL2248187 0.74 GBA1 (0.48)
SCHEMBL9311027 0.70 HTR6 (0.75) HTR6ESR1ESR2SLC22A1PRCP
SCHEMBL2242306 0.69 ALDH1A1 (0.49) KDM4ENPC1ALDH1A1LMNAGLA
SCHEMBL22606737 0.69 HTR6 (0.55) HTR6ESR1ESR2MTNR1AMTNR1B
SCHEMBL2245636 0.69 GBA1 (0.44) HTR6KDM4ENPC1ALDH1A1LMNA
SCHEMBL27579440 0.68 HTR6 (0.51) HTR6IDO1
SCHEMBL2243951 0.68 IDO1 (0.40) KDM4ENPC1ALDH1A1LMNAGLA
SCHEMBL27780844 0.68 GBA1 (0.50) KDM4ENPC1ALDH1A1LMNAGLA
SCHEMBL1615946 0.66 GBA1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099763-B1 2-AMINOQUINOLINES AS 5-HT(5A) RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-08-11 EP disclosed