SCHEMBL29062471

SCHEMBL29062471

O=c1[nH]c(Nc2ccccn2)nc2c1nc(-c1ccc([N+](=O)[O-])nc1)n2C1=CCCCC1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UGT1A1 P22309 1/20 0.33
MAT2A P31153 1/20 0.33
SLCO1B1 Q9Y6L6 1/20 0.33
PDE9A O76083 1/20 0.31
MEN1 O00255 2/20 0.30
NPC1 O15118 2/20 0.30
RAB9A P51151 2/20 0.30
KMT2A Q03164 2/20 0.30
KDM4E B2RXH2 1/20 0.30
TDP2 O95551 1/20 0.30
HSP90AA1 P07900 1/20 0.30
MAPT P10636 1/20 0.30
MAPK1 P28482 1/20 0.30
CASP3 P42574 1/20 0.30
BLM P54132 1/20 0.30
CASP7 P55210 1/20 0.30
CASP9 P55211 1/20 0.30
CASP6 P55212 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
PIM1 P11309 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30584032 1.00 UGT1A1 (0.33) UGT1A1MAT2ASLCO1B1PDE9AMEN1
SCHEMBL30584014 0.79 MAT2A (0.41) UGT1A1MAT2ASLCO1B1MEN1NPC1
SCHEMBL29062470 0.79 MAT2A (0.41) UGT1A1MAT2ASLCO1B1MEN1NPC1
SCHEMBL30584019 0.79 MAT2A (0.41) UGT1A1MAT2ASLCO1B1MEN1NPC1
SCHEMBL30584023 0.78 UGT1A1 (0.33) UGT1A1MAT2ASLCO1B1
SCHEMBL29062443 0.75 PIM1 (0.36) UGT1A1MAT2ASLCO1B1MEN1NPC1
SCHEMBL30719375 0.74 PIM1 (0.40) MEN1NPC1RAB9AKMT2AKDM4E
SCHEMBL30584033 0.73 MAPT (0.31) MAPT
SCHEMBL29062469 0.73 MAPT (0.31) MAPT
SCHEMBL29062438 0.67 MAT2A (0.43) UGT1A1MAT2ASLCO1B1MEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117777134-A Polycyclic compounds as MAT2A inhibitors 艾立康药业股份有限公司 2024-03-29 CN disclosed
CN-116425751-B Polycyclic compounds as MAT2A inhibitors 艾立康药业股份有限公司 2024-01-23 CN disclosed
CN-116425751-A Polycyclic compounds as MAT2A inhibitors 艾立康药业股份有限公司 2023-07-14 CN disclosed