SCHEMBL29065385

SCHEMBL29065385

C#Cn1nnc(-c2cccc(Br)c2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.42
NPC1 O15118 6/20 0.38
RAB9A P51151 6/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
TSHR P16473 2/20 0.38
TP53 P04637 1/20 0.38
KMT2A Q03164 5/20 0.38
ALDH1A1 P00352 4/20 0.38
MEN1 O00255 4/20 0.38
MAPT P10636 2/20 0.38
HPGD P15428 2/20 0.38
HTT P42858 1/20 0.38
IDO1 P14902 1/20 0.37
METAP2 P50579 1/20 0.37
CYP1A2 P05177 1/20 0.37
HCRTR1 O43613 1/20 0.37
CASP3 P42574 1/20 0.37
SENP8 Q96LD8 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1092403 0.76 AHR (0.45) AHRNPC1RAB9ASMN1; SMN2TSHR
SCHEMBL27628842 0.73 AHR (0.43) AHRNPC1RAB9ASMN1; SMN2TSHR
SCHEMBL13947009 0.73 SMN1; SMN2 (0.53) AHRNPC1RAB9ASMN1; SMN2TSHR
SCHEMBL7017606 0.72 SMN1; SMN2 (0.43) AHRNPC1RAB9ASMN1; SMN2TSHR
SCHEMBL13863817 0.72 AAK1 (0.47) AHRNPC1RAB9AGABRG2GABRB3
SCHEMBL4639604 0.69 RAB9A (0.42) AHRNPC1RAB9ASMN1; SMN2TSHR
SCHEMBL4700157 0.68 GRM5 (0.67) NPC1RAB9ATP53
SCHEMBL4547022 0.67 RAB9A (0.56) AHRNPC1RAB9ASMN1; SMN2TSHR
SCHEMBL29878444 0.67 RAB9A (0.56) AHRNPC1RAB9ASMN1; SMN2TSHR
SCHEMBL6188523 0.67 RAB9A (0.55) NPC1RAB9ASMN1; SMN2TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116675684-B Alkynyl-containing condensed ring derivative antagonist, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-11-07 CN disclosed
CN-116675684-A Alkynyl-containing condensed ring derivative antagonist, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-09-01 CN disclosed