SCHEMBL29068286

SCHEMBL29068286

COc1cccc(CNCc2c(C(=O)O)n(Cc3ccc(C)cc3)c3cc(C(C)C)ccc23)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
YWHAH Q04917 6/20 1.00
KCNH2 Q12809 1/20 1.00
TP53 P04637 11/20 0.81
POLB P06746 2/20 0.63
MAPT P10636 2/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30490434 0.93 YWHAH (0.90) YWHAHKCNH2TP53POLBMAPT
SCHEMBL30490432 0.93 YWHAH (1.00) YWHAHKCNH2TP53POLBMAPT
SCHEMBL30490431 0.87 TP53 (0.91) YWHAHKCNH2TP53POLBMAPT
SCHEMBL30490429 0.86 YWHAH (1.00) YWHAHKCNH2TP53POLBMAPT
SCHEMBL30490428 0.84 YWHAH (0.79) YWHAHKCNH2TP53POLBMAPT
SCHEMBL30490436 0.81 TP53 (0.77) YWHAHKCNH2TP53POLBMAPT
SCHEMBL30490435 0.74 TP53 (0.73) YWHAHKCNH2TP53POLBMAPT
SCHEMBL2555312 0.70 TP53 (0.59) YWHAHKCNH2TP53POLBMAPT
SCHEMBL29845649 0.70 TP53 (0.87) YWHAHTP53POLBMAPT
SCHEMBL29845533 0.69 TP53 (0.84) YWHAHTP53POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116554080-A 1H-indole-2-carboxylic acid derivative, pharmaceutical composition and application 深圳市坤健创新药物研究院 2023-08-08 CN disclosed