SCHEMBL30490432

SCHEMBL30490432

COc1cccc(CNCc2c(C(=O)O)n(Cc3ccc(O)cc3)c3cc(C(C)C)ccc23)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
YWHAH Q04917 6/20 1.00
KCNH2 Q12809 1/20 0.87
TP53 P04637 10/20 0.72
MAPT P10636 2/20 0.61
POLB P06746 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29068286 0.93 YWHAH (1.00) YWHAHKCNH2TP53MAPTPOLB
SCHEMBL30490434 0.93 YWHAH (0.90) YWHAHKCNH2TP53MAPTPOLB
SCHEMBL30490431 0.89 TP53 (0.91) YWHAHKCNH2TP53MAPTPOLB
SCHEMBL30490429 0.86 YWHAH (1.00) YWHAHKCNH2TP53MAPTPOLB
SCHEMBL30490428 0.85 YWHAH (0.79) YWHAHKCNH2TP53MAPTPOLB
SCHEMBL30490436 0.81 TP53 (0.77) YWHAHKCNH2TP53MAPTPOLB
SCHEMBL29845533 0.69 TP53 (0.84) YWHAHTP53MAPTPOLB
SCHEMBL30490435 0.69 TP53 (0.73) YWHAHKCNH2TP53MAPTPOLB
SCHEMBL29845629 0.68 MAPT (0.86) YWHAHTP53MAPTPOLB
SCHEMBL29845627 0.68 MAPT (0.86) YWHAHTP53MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116554080-A 1H-indole-2-carboxylic acid derivative, pharmaceutical composition and application 深圳市坤健创新药物研究院 2023-08-08 CN disclosed