SCHEMBL3721157

SCHEMBL3721157

COC(=O)c1cc(NCc2ccccc2)nc(-c2ccc(C#Cc3cccnc3)cc2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.48
ABCG2 Q9UNQ0 3/20 0.48
ABCC1 P33527 1/20 0.48
PTGS2 P35354 5/20 0.44
CYP1A2 P05177 6/20 0.43
CYP3A4 P08684 6/20 0.43
CYP2D6 P10635 5/20 0.43
CLK4 Q9HAZ1 4/20 0.43
USP2 O75604 2/20 0.43
CYP2C19 P33261 2/20 0.43
HPGD P15428 2/20 0.43
PTGES O14684 1/20 0.42
FFAR1 O14842 1/20 0.42
ALDH1A1 P00352 3/20 0.41
MAPK1 P28482 1/20 0.41
HSD17B10 Q99714 3/20 0.41
ALOX15 P16050 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
HIF1A Q16665 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13188295 0.88 ABCB1 (0.48) ABCB1ABCG2ABCC1PTGS2CYP1A2
SCHEMBL3718011 0.86 FGFR4 (0.40) CYP1A2CYP3A4CLK4CYP2C19FFAR1
SCHEMBL3710406 0.85 PIK3CA (0.46) ABCB1ABCG2ABCC1CYP1A2CYP3A4
SCHEMBL3713514 0.84 FPR2 (0.40) PTGESFFAR1ALDH1A1ACACB
SCHEMBL3714572 0.80 P2RY12 (0.46) CYP1A2CYP3A4CYP2D6CLK4CYP2C19
SCHEMBL3711805 0.78 CYP19A1 (0.49) ABCG2FFAR1ALDH1A1
SCHEMBL13188297 0.78 P2RY12 (0.40) CYP1A2CYP3A4CLK4FFAR1ALDH1A1
SCHEMBL3713214 0.78 CLK4 (0.48) CYP1A2CYP3A4CYP2D6CLK4CYP2C19
SCHEMBL3710041 0.77 HDAC1 (0.46) ABCB1ABCG2ABCC1CYP1A2CYP3A4
SCHEMBL2907007 0.76 ABCB1 (0.58) ABCB1ABCG2ABCC1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed