SCHEMBL2907018

SCHEMBL2907018

O=C(O)c1cc(OC2CNC2)cc(-c2ccccc2)n1

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 10/20 0.50
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
P2RY12 Q9H244 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL317418 0.85 MCL1 (0.51) MCL1P2RY12
SCHEMBL1201785 0.80 GRM5 (0.50) MCL1P2RY12
SCHEMBL1111184 0.76 MCL1 (0.64) MCL1KDM4EALDH1A1
SCHEMBL986309 0.76 USP30 (0.47) MCL1P2RY12
SCHEMBL2907048 0.73 P2RY12 (0.43) MCL1P2RY12
SCHEMBL4271936 0.72 NPC1 (0.55) MCL1KDM4EALDH1A1P2RY12
SCHEMBL4265711 0.71 MCL1 (0.74) MCL1P2RY12
SCHEMBL2899930 0.70 MCL1 (0.52) MCL1KDM4EALDH1A1
SCHEMBL2906146 0.70 ALDH1A1 (0.52) MCL1KDM4EALDH1A1P2RY12
Oxalic Acid SCHEMBL9595892 0.70 SLC6A4 (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2217606-A1 SOLUBILIZED THIAZOLOPYRIDINES Sirtris Pharmaceuticals, Inc. (US) 2010-08-18 EP disclosed
WO-2009061453-A1 SOLUBILIZED THIAZOLOPYRIDINES SIRTRIS PHARMACEUTICALS, INC. (US) 2009-05-14 WO disclosed