SCHEMBL29074142

SCHEMBL29074142

Nc1ccc(Br)c(N2CCC(F)(F)CC2)n1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MBOAT4 Q96T53 6/20 0.49
PIK3CA P42336 1/20 0.39
MTOR P42345 1/20 0.39
NOS3 P29474 2/20 0.35
NOS1 P29475 2/20 0.35
NOS2 P35228 2/20 0.35
FFAR2 O15552 5/20 0.35
SCN10A Q9Y5Y9 4/20 0.35
MAOB P27338 1/20 0.34
PDE10A Q9Y233 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30527887 1.00 MBOAT4 (0.49) MBOAT4PIK3CAMTORNOS3NOS1
SCHEMBL26151136 0.83 PIK3CA (0.41) MBOAT4PIK3CAMTORNOS3NOS1
SCHEMBL30788625 0.82 IDH1 (0.41) MBOAT4PIK3CAMTORNOS3NOS1
SCHEMBL26883498 0.82 IDH1 (0.41) MBOAT4PIK3CAMTORNOS3NOS1
SCHEMBL22122604 0.81 PIK3CA (0.42) MBOAT4PIK3CAMTORNOS3NOS1
SCHEMBL26151845 0.78 FFAR2 (0.38) PIK3CAMTORFFAR2
SCHEMBL26151146 0.77 WHR1 (0.45) MBOAT4PIK3CAMTORNOS3NOS1
SCHEMBL22122552 0.77 MBOAT4 (0.44) MBOAT4PIK3CAMTORNOS3NOS1
SCHEMBL29074131 0.76 PIK3CA (0.39) MBOAT4PIK3CAMTORNOS3NOS1
SCHEMBL29074141 0.75 FFAR2 (0.41) PIK3CAMTORNOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116554151-B Kinesin KIF18A inhibitor and application thereof 上海湃隆生物科技有限公司 2024-09-20 CN disclosed
CN-116554151-A Kinesin KIF18A inhibitor and application thereof 上海湃隆生物科技有限公司 2023-08-08 CN disclosed