SCHEMBL2907443

SCHEMBL2907443

NC(=O)COc1ccccc1-c1nc2ccccc2n1Cc1c(F)cccc1Cl

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.54
MAPT P10636 2/20 0.54
ALDH1A1 P00352 2/20 0.53
NPSR1 Q6W5P4 2/20 0.53
GAA P10253 1/20 0.53
RECQL P46063 1/20 0.53
THRB P10828 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
KCNN4 O15554 1/20 0.43
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
PLA2G2A P14555 2/20 0.42
PDE6D O43924 2/20 0.42
KMT2A Q03164 1/20 0.41
CDK1 P06493 1/20 0.41
CDK4 P11802 1/20 0.41
CDK2 P24941 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2909757 0.93 KCNN4 (0.47) TP53MAPTALDH1A1NPSR1GAA
SCHEMBL2906933 0.90 NPSR1 (0.53) TP53MAPTALDH1A1NPSR1GAA
SCHEMBL638894 0.87 NPSR1 (0.48) TP53MAPTALDH1A1NPSR1GAA
SCHEMBL639847 0.84 KDM4E (0.50) MAPTALDH1A1NPSR1GAARECQL
SCHEMBL638902 0.84 NPSR1 (0.48) TP53MAPTALDH1A1NPSR1GAA
SCHEMBL639087 0.83 NPSR1 (0.47) TP53MAPTALDH1A1NPSR1GAA
SCHEMBL641038 0.83 KDM4E (0.56) TP53MAPTALDH1A1NPSR1SMN1; SMN2
SCHEMBL2907639 0.79 PLA2G2A (0.44) TP53MAPTALDH1A1NPSR1GAA
SCHEMBL2907759 0.79 PLA2G2A (0.43) TP53MAPTALDH1A1GAASMN1; SMN2
SCHEMBL2903474 0.79 KMT2A (0.42) TP53MAPTALDH1A1NPSR1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121627-B1 BENZIMIDAZOLE DERIVATIVES MERCK PATENT GMBH (DE) 2010-08-18 EP claimed