SCHEMBL2907904

SCHEMBL2907904

CCOc1cc2nc(CC)c(C(=O)O)c(Nc3cc(C)ccc3F)c2cc1N1CCN(C(C)C)CC1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.50
SCN5A Q14524 11/20 0.50
CSF1R P07333 5/20 0.44
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2914186 0.89 KCNH2 (0.57) KCNH2SCN5ACSF1R
SCHEMBL2907901 0.82 KCNH2 (0.63) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL1276767 0.82 KCNH2 (0.74) KCNH2SCN5ACSF1R
SCHEMBL2911894 0.79 SCN5A (0.65) KCNH2SCN5ACSF1R
SCHEMBL2907902 0.78 KCNH2 (0.54) KCNH2SCN5ACSF1R
SCHEMBL2909211 0.78 CSF1R (0.51) KCNH2SCN5ACSF1R
SCHEMBL2910575 0.77 KCNH2 (0.68) KCNH2SCN5ACSF1R
SCHEMBL2914061 0.77 CSF1R (0.49) KCNH2SCN5ACSF1R
SCHEMBL2911756 0.77 KCNH2 (0.68) KCNH2SCN5ACSF1R
SCHEMBL2911555 0.77 KCNH2 (0.53) KCNH2SCN5ACSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed