SCHEMBL29079141

SCHEMBL29079141

COC(=O)C(NC(=O)OC(C)(C)C)C(C)Oc1ccc(Br)cc1N

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 17/20 0.47
KLK5 Q9Y337 1/20 0.37
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29079186 0.90 AAK1 (0.47) AAK1CTSSCTSK
SCHEMBL29079137 0.83 AAK1 (0.42) AAK1ALDH1A1MAPT
SCHEMBL29079182 0.81 AAK1 (0.47) AAK1ALDH1A1MAPTCTSSCTSK
SCHEMBL27534635 0.76 TRPA1 (0.40) AAK1CTSSCTSK
SCHEMBL8905741 0.76 TRPA1 (0.40) AAK1CTSSCTSK
SCHEMBL8905745 0.76 TRPA1 (0.40) AAK1CTSSCTSK
SCHEMBL1562328 0.76 TRPA1 (0.40) AAK1CTSSCTSK
SCHEMBL1562711 0.75 PPARG (0.41) AAK1ALDH1A1MAPT
SCHEMBL22525379 0.74 CACNA1B (0.48) AAK1KLK5ALDH1A1MAPTCTSS
SCHEMBL25076071 0.73 KLK5 (0.49) KLK5CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116640156-A RIPK1 inhibitors 上海齐鲁制药研究中心有限公司 2023-08-25 CN disclosed