SCHEMBL29079137

SCHEMBL29079137

COC(=O)C(NC(=O)OC(C)(C)C)C(C)Oc1ccc(Br)cc1[N+](=O)[O-]

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 11/20 0.42
GSTP1 P09211 1/20 0.40
GSTM2 P28161 1/20 0.40
PDK1 Q15118 1/20 0.37
ALDH1A1 P00352 3/20 0.37
ABCB1 P08183 1/20 0.37
ABCC1 P33527 1/20 0.37
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29079146 0.91 AAK1 (0.43) AAK1PDK1ALDH1A1MAPT
SCHEMBL29079141 0.83 AAK1 (0.47) AAK1ALDH1A1MAPT
SCHEMBL29079144 0.82 AAK1 (0.43) AAK1GSTP1GSTM2ALDH1A1GAA
SCHEMBL8904841 0.78 ALDH1A1 (0.40) AAK1PDK1ALDH1A1GAAMAPT
SCHEMBL27391920 0.78 ALDH1A1 (0.40) AAK1PDK1ALDH1A1GAAMAPT
SCHEMBL8904838 0.78 ALDH1A1 (0.40) AAK1PDK1ALDH1A1GAAMAPT
SCHEMBL1561567 0.78 ALDH1A1 (0.40) AAK1PDK1ALDH1A1GAAMAPT
SCHEMBL16851396 0.78 PDK1 (0.46) PDK1ALDH1A1ABCB1ABCC1MAPT
SCHEMBL531814 0.78 PDK1 (0.46) PDK1ALDH1A1ABCB1ABCC1MAPT
SCHEMBL1561729 0.77 MAPT (0.53) ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116640156-A RIPK1 inhibitors 上海齐鲁制药研究中心有限公司 2023-08-25 CN disclosed