SCHEMBL29079760

SCHEMBL29079760

COC(=O)c1ccc2ncn(CC3CCO3)c2n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.40
GAA P10253 6/20 0.40
KDM4E B2RXH2 6/20 0.40
HPGD P15428 3/20 0.40
HTT P42858 1/20 0.40
TSHR P16473 3/20 0.37
NPSR1 Q6W5P4 1/20 0.37
KMT2A Q03164 3/20 0.37
MAPK1 P28482 2/20 0.36
MEN1 O00255 2/20 0.35
RAB9A P51151 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
ESR1 P03372 1/20 0.35
MAPT P10636 1/20 0.35
GLA P06280 4/20 0.35
CASP1 P29466 2/20 0.35
CASP7 P55210 2/20 0.35
HSD17B10 Q99714 2/20 0.35
TRPA1 O75762 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29079758 1.00 ALDH1A1 (0.40) ALDH1A1GAAKDM4EHPGDHTT
SCHEMBL29558931 1.00 ALDH1A1 (0.40) ALDH1A1GAAKDM4EHPGDHTT
SCHEMBL25435833 0.89 CYP1A2 (0.40) ALDH1A1GAAKDM4EHPGDHTT
SCHEMBL29668753 0.89 CYP1A2 (0.40) ALDH1A1GAAKDM4EHPGDHTT
SCHEMBL30124865 0.89 CYP1A2 (0.40) ALDH1A1GAAKDM4EHPGDHTT
SCHEMBL30149437 0.88 ALDH1A1 (0.46) ALDH1A1GAAKDM4EHPGDHTT
SCHEMBL30174413 0.88 ALDH1A1 (0.46) ALDH1A1GAAKDM4EHPGDHTT
SCHEMBL25405514 0.86 GLP1R (0.41) ALDH1A1GAAKDM4EHPGDHTT
SCHEMBL25405520 0.86 GLP1R (0.41) ALDH1A1GAAKDM4EHPGDHTT
SCHEMBL29480771 0.86 TRPA1 (0.40) ALDH1A1GAAKDM4EHPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024046342-A1 BENZO BICYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, AND USE THEREOF 广州市联瑞制药有限公司 2024-03-07 WO disclosed
CN-117355517-A Macrocyclic glucagon-like peptide 1 receptor agonists 伊莱利利公司 2024-01-05 CN disclosed
CN-114728939-B GLP-1 receptor agonists and uses thereof 日东制药株式会社 2023-12-08 CN disclosed
WO-2023169436-A1 BENZO BICYCLIC COMPOUND, AND PREPARATION METHOD AND APPLICATION THEREOF 广州市联瑞制药有限公司 2023-09-14 WO disclosed
CN-116406360-A Heterocyclic GLP-1 agonists 加舒布鲁姆生物公司 2023-07-07 CN disclosed
CN-116348464-A Benzimidazolone GLP-1 receptor agonists and uses thereof 杭州中美华东制药有限公司 2023-06-27 CN disclosed
CN-115697999-A Heterocyclic GLP-1 agonists 加舒布鲁姆生物公司 2023-02-03 CN disclosed
CN-115515956-A Benzimidazole derivative and preparation method and medical application thereof 深圳信立泰药业股份有限公司 2022-12-23 CN disclosed
CN-114728939-A GLP-1 receptor agonists and uses thereof 日东制药株式会社 2022-07-08 CN disclosed
CN-113480534-B Benzimidazole or azabenzimidazole-6-carboxylic acid compounds and application thereof 广州必贝特医药股份有限公司 2022-05-13 CN disclosed
WO-2022068772-A1 BENZIMIDAZOLE DERIVATIVE, AND PREPARATION METHOD THEREFOR, AND MEDICAL USE THEREOF 深圳信立泰药业股份有限公司 2022-04-07 WO disclosed