SCHEMBL29084385

SCHEMBL29084385

O=Cc1ccccc1C(=O)c1cccc(F)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.50
CES1 P23141 2/20 0.50
PARP1 P09874 1/20 0.47
NPC1 O15118 4/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
HPGD P15428 3/20 0.47
MAPT P10636 2/20 0.47
HTT P42858 2/20 0.47
LMNA P02545 2/20 0.47
KDM4E B2RXH2 1/20 0.47
TSHR P16473 1/20 0.47
ALOX12 P18054 1/20 0.47
HDAC1 Q13547 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
RAB9A P51151 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
CTNNB1 P35222 1/20 0.43
WNT3A P56704 1/20 0.43
BDKRB1 P46663 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12295978 0.82 FASN (0.49) PARP1NPC1MEN1KMT2AKDM4E
SCHEMBL24176082 0.82 UNG (0.56) MEN1KMT2AMAPTLMNAHDAC1
SCHEMBL28376319 0.81 NPC1 (0.44) CES2CES1NPC1MEN1KMT2A
SCHEMBL1004343 0.81 AKR1C3 (0.57) MEN1KMT2AMAPTLMNAKDM4E
SCHEMBL1513045 0.80 CES2 (0.57) CES2CES1PARP1NPC1MEN1
SCHEMBL10321851 0.79 LMNA (0.44) MEN1KMT2AMAPTLMNASMN1; SMN2
SCHEMBL28376318 0.79 MAPK1 (0.44) NPC1MEN1KMT2AMAPTHTT
SCHEMBL10997315 0.78 AKR1C3 (0.66) CES2CES1PARP1NPC1MEN1
SCHEMBL8022367 0.77 CES2 (0.53) CES2CES1PARP1NPC1MEN1
SCHEMBL29963651 0.77 MAPT (0.65) CES2CES1PARP1NPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117285512-A 2, 5-diketopiperazine-imidazole compound, preparation method and application thereof 大连万众益生大健康有限公司 2023-12-26 CN disclosed
CN-114685456-B 2, 5-diketopiperazine compound derivative, preparation method thereof, pharmaceutical composition and application thereof 大连万众益生大健康有限公司 2023-10-10 CN disclosed