SCHEMBL29084871

SCHEMBL29084871

NC(=O)N1CCc2cc(-c3ccccc3)ccc2C1c1c[nH]c2ncc(F)cc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 3/20 0.40
AXL P30530 8/20 0.39
AURKA O14965 2/20 0.39
SGK2 Q9HBY8 2/20 0.39
CDC7 O00311 1/20 0.39
PLK4 O00444 1/20 0.39
CHEK1 O14757 1/20 0.39
MAPK13 O15264 1/20 0.39
PDPK1 O15530 1/20 0.39
DYRK3 O43781 1/20 0.39
ROCK2 O75116 1/20 0.39
RPS6KA5 O75582 1/20 0.39
PRKD3 O94806 1/20 0.39
PAK4 O96013 1/20 0.39
CHEK2 O96017 1/20 0.39
ABL1 P00519 1/20 0.39
EGFR P00533 1/20 0.39
NTRK1 P04629 1/20 0.39
INSR P06213 1/20 0.39
LCK P06239 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30593275 1.00 HSD11B1 (0.40) HSD11B1AXLAURKASGK2CDC7
SCHEMBL29084879 0.89 AURKA (0.43) HSD11B1AXLAURKASGK2CDC7
SCHEMBL29084845 0.89 JAK2 (0.43) HSD11B1AXLAURKASGK2CDC7
SCHEMBL30593219 0.89 AURKA (0.43) HSD11B1AXLAURKASGK2CDC7
SCHEMBL30593241 0.89 JAK2 (0.43) HSD11B1AXLAURKASGK2CDC7
SCHEMBL30593317 0.84 HSD11B1 (0.43) HSD11B1ESR1ESR2
SCHEMBL30593229 0.81 ESR1 (0.39) HSD11B1ESR1ESR2
SCHEMBL30593227 0.81 ECE1 (0.44) HSD11B1ESR1ESR2
SCHEMBL29084778 0.79 MAP2 (0.40) HSD11B1PRKAA1ESR1ESR2
SCHEMBL30593278 0.79 MAP2 (0.40) HSD11B1PRKAA1ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116789641-A Dihydro isoquinoline compound and medical application thereof 中国科学院上海药物研究所 2023-09-22 CN disclosed