SCHEMBL30593241

SCHEMBL30593241

NC(=O)N1CCc2cc(-c3ccccc3)ccc2C1c1c[nH]c2ncc(Cl)cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.43
PAK1 Q13153 4/20 0.42
PKN1 Q16512 1/20 0.42
MAP2 P11137 1/20 0.40
HSD11B1 P28845 2/20 0.40
AXL P30530 4/20 0.39
SGK2 Q9HBY8 3/20 0.39
PRKD3 O94806 2/20 0.39
EGFR P00533 2/20 0.39
NTRK1 P04629 2/20 0.39
LCK P06239 2/20 0.39
FYN P06241 2/20 0.39
FLT4 P35916 2/20 0.39
KDR P35968 2/20 0.39
FLT3 P36888 2/20 0.39
FRK P42685 2/20 0.39
CLK2 P49760 2/20 0.39
CAMK2B Q13554 2/20 0.39
CAMK2G Q13555 2/20 0.39
CAMK2D Q13557 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29084845 1.00 JAK2 (0.43) JAK2PAK1PKN1MAP2HSD11B1
SCHEMBL30593275 0.89 HSD11B1 (0.40) PAK1PKN1HSD11B1AXLSGK2
SCHEMBL29084879 0.89 AURKA (0.43) JAK2PAK1PKN1HSD11B1AXL
SCHEMBL29084871 0.89 HSD11B1 (0.40) PAK1PKN1HSD11B1AXLSGK2
SCHEMBL30593219 0.89 AURKA (0.43) JAK2PAK1PKN1HSD11B1AXL
SCHEMBL31083748 0.86 KIF11 (0.48) MAP2HSD11B1KIF11ESR1ESR2
SCHEMBL30593227 0.83 ECE1 (0.44) HSD11B1KIF11ESR1ESR2
SCHEMBL29084778 0.80 MAP2 (0.40) MAP2HSD11B1PRKAA1KIF11ESR1
SCHEMBL30593278 0.80 MAP2 (0.40) MAP2HSD11B1PRKAA1KIF11ESR1
SCHEMBL30593229 0.80 ESR1 (0.39) HSD11B1KIF11ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118742543-A Dihydro isoquinoline compound and medical application thereof 中国科学院上海药物研究所 2024-10-01 CN disclosed
CN-116789641-A Dihydro isoquinoline compound and medical application thereof 中国科学院上海药物研究所 2023-09-22 CN disclosed