SCHEMBL29101367

SCHEMBL29101367

CCCCC(OC(N)=O)C(=O)Nc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.54
ALDH1A1 P00352 2/20 0.54
KMT2A Q03164 2/20 0.54
MAPT P10636 1/20 0.54
MAPK1 P28482 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
HDAC2 Q92769 8/20 0.53
KLK7 P49862 4/20 0.51
HDAC8 Q9BY41 6/20 0.47
HDAC3 O15379 5/20 0.47
HDAC6 Q9UBN7 5/20 0.47
HDAC1 Q13547 4/20 0.47
HDAC4 P56524 2/20 0.47
HDAC7 Q8WUI4 2/20 0.47
HDAC10 Q969S8 2/20 0.47
HDAC11 Q96DB2 2/20 0.47
HDAC9 Q9UKV0 2/20 0.47
HDAC5 Q9UQL6 2/20 0.47
HSD17B10 Q99714 1/20 0.47
NPSR1 Q6W5P4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29101361 0.86 KLK7 (0.50) MEN1ALDH1A1KMT2AMAPTMAPK1
SCHEMBL3955546 0.86 HDAC2 (0.51) MEN1ALDH1A1KMT2AMAPTMAPK1
SCHEMBL11636534 0.82 HDAC2 (0.56) MEN1ALDH1A1KMT2AMAPTMAPK1
SCHEMBL3960647 0.81 SIRT1 (0.59) HDAC2KLK7
SCHEMBL29383934 0.80 KCNH2 (0.45) MEN1ALDH1A1KMT2AMAPTMAPK1
SCHEMBL5264997 0.78 MEN1 (0.61) MEN1ALDH1A1KMT2AMAPTMAPK1
SCHEMBL9267426 0.78 MEN1 (0.61) MEN1ALDH1A1KMT2AMAPTMAPK1
SCHEMBL11642274 0.78 HDAC2 (0.62) MEN1ALDH1A1KMT2AMAPTMAPK1
SCHEMBL7099035 0.77 MEN1 (0.78) MEN1ALDH1A1KMT2AMAPTMAPK1
SCHEMBL11644668 0.77 HDAC2 (0.68) MEN1ALDH1A1KMT2AMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114761079-B Benzothiazepine compounds and their use as bile acid modulators 阿尔比里奥公司 2024-05-28 CN disclosed
CN-117412955-A Benzothiazepine compounds and their use as bile acid modulators 阿尔比里奥公司 2024-01-16 CN disclosed
CN-116583504-A Benzothiazepine compounds and their use as bile acid modulators 阿尔比里奥公司 2023-08-11 CN disclosed