SCHEMBL2910148

SCHEMBL2910148

CCOC(=O)c1cnc2cc(OCC)c(N3CCCN(C)CC3)cc2c1Nc1cccc(Cl)c1C

nearest known ligand 0.69

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.69
SCN5A Q14524 3/20 0.69
CSF1R P07333 11/20 0.57
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
GAA P10253 2/20 0.48
SLC2A1 P11166 1/20 0.48
MAPK10 P53779 1/20 0.47
MAPT P10636 2/20 0.46
THRB P10828 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2910208 0.97 KCNH2 (0.73) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2913553 0.94 KCNH2 (0.79) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2911736 0.92 KCNH2 (0.81) KCNH2SCN5ACSF1R
SCHEMBL2912865 0.92 KCNH2 (0.67) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2905267 0.92 KCNH2 (0.65) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2912423 0.91 KCNH2 (0.84) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2912268 0.90 KCNH2 (0.63) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2911553 0.90 KCNH2 (0.67) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2909672 0.89 KCNH2 (0.71) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2914208 0.89 KCNH2 (0.86) KCNH2SCN5ACSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed