SCHEMBL2912865

SCHEMBL2912865

CCOC(=O)c1cnc2cc(OCC)c(N3CCCN(C)CC3)cc2c1Nc1cccc(F)c1C

nearest known ligand 0.67

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 9/20 0.67
SCN5A Q14524 4/20 0.63
CSF1R P07333 9/20 0.62
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
GAA P10253 1/20 0.48
SLC2A1 P11166 1/20 0.48
MAPT P10636 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2907886 0.97 KCNH2 (0.67) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2905878 0.93 KCNH2 (0.78) KCNH2SCN5ACSF1R
SCHEMBL2910148 0.92 KCNH2 (0.69) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2910961 0.91 KCNH2 (0.67) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2913889 0.90 KCNH2 (0.57) KCNH2SCN5ACSF1RMAPT
SCHEMBL2911163 0.89 KCNH2 (0.73) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2909951 0.89 KCNH2 (0.79) KCNH2SCN5ACSF1R
SCHEMBL2911553 0.89 KCNH2 (0.67) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2913052 0.89 KCNH2 (0.71) KCNH2SCN5ACSF1RMEN1KMT2A
SCHEMBL2905342 0.89 KCNH2 (0.84) KCNH2SCN5ACSF1RMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed