SCHEMBL2910443

SCHEMBL2910443

COC1CC(=O)CCc2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.43
CYP2A6 P11509 1/20 0.41
ACP3 P15309 1/20 0.40
SRD5A1 P18405 2/20 0.39
RET P07949 1/20 0.38
HTR2A P28223 1/20 0.38
CETP P11597 1/20 0.37
PIN1 Q13526 1/20 0.36
PDPK1 O15530 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GID4 Q8IVV7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24140334 0.84 IDO1 (0.47) IDO1ACP3RETHTR2ACETP
SCHEMBL16866695 0.79 IDO1 (0.44) IDO1
SCHEMBL18959593 0.79 IDO1 (0.44) IDO1
SCHEMBL2907549 0.79 CA9 (0.38) HTR2AKDM4EALDH1A1
SCHEMBL447420 0.76 IDO1 (0.66) IDO1PIN1PDPK1
SCHEMBL21300294 0.76 IDO1 (0.66) IDO1PIN1PDPK1
SCHEMBL14209228 0.76 IDO1 (0.66) IDO1PIN1PDPK1
SCHEMBL3814265 0.75 IDO1 (0.46) IDO1CYP2A6SRD5A1HTR2APIN1
SCHEMBL2910014 0.74 PNMT (0.42) HTR2AALDH1A1SMN1; SMN2
SCHEMBL2472307 0.73 IDO1 (0.68) IDO1PDPK1KDM4EGID4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222647-A1 FUSED BICYCLIC DERIVATIVES OF 2,4-DIAMINOPYRIMIDINE AS ALK AND C-MET INHIBITORS Cephalon, Inc. (US) 2010-09-01 EP disclosed
WO-2008051547-A1 FUSED BICYCLIC DERIVATIVES OF 2,4-DIAMINOPYRIMIDINE AS ALK AND C-MET INHIBITORS CEPHALON, INC. (US) 2008-05-02 WO disclosed