SCHEMBL2910776

SCHEMBL2910776

Nc1nc(NCCCn2cc(C(=O)O)c(-c3ccc(C(F)(F)F)cc3F)c2)ccc1[N+](=O)[O-]

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.37
HTT P42858 3/20 0.37
GAA P10253 2/20 0.37
AKR1B1 P15121 1/20 0.37
AKR1C4 P17516 1/20 0.37
AKR1C3 P42330 1/20 0.37
AKR1C2 P52895 1/20 0.37
AKR1C1 Q04828 1/20 0.37
SERPINE1 P05121 2/20 0.37
RAB9A P51151 1/20 0.36
GSK3B P49841 4/20 0.36
GSK3A P49840 3/20 0.36
EIF4E P06730 3/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
LMNA P02545 1/20 0.34
THRB P10828 1/20 0.34
CDK1 P06493 2/20 0.34
TTR P02766 1/20 0.34
PPOX P50336 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2912304 0.90 GSK3B (0.38) MAPTHTTGSK3BGSK3AEIF4E
SCHEMBL2909502 0.90 GSK3B (0.35) MAPTHTTGAASERPINE1RAB9A
SCHEMBL2906807 0.89 GSK3B (0.45) MAPTGSK3BGSK3AEIF4ELMNA
SCHEMBL2908029 0.89 GSK3B (0.37) AKR1C2AKR1C1GSK3BGSK3AEIF4E
SCHEMBL2911406 0.89 EIF4E (0.37) MAPTHTTGAAAKR1B1AKR1C4
SCHEMBL2904400 0.88 ALOX5AP (0.43) MAPTHTTGAARAB9AGSK3B
SCHEMBL2912014 0.88 ALOX5AP (0.43) MAPTHTTGAARAB9AGSK3B
SCHEMBL2909381 0.88 MAPT (0.38) MAPTHTTGAASERPINE1RAB9A
SCHEMBL2907210 0.88 MAPT (0.38) MAPTHTTGAASERPINE1RAB9A
SCHEMBL2906887 0.84 GSK3B (0.43) HTTGSK3BGSK3AEIF4ECDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-B1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 NOVARTIS VACCINES & DIAGNOSTIC (US) 2010-08-11 EP disclosed