SCHEMBL2911121

SCHEMBL2911121

C[C@@H](O)CNC(=O)c1cn(CCCNc2ccc([N+](=O)[O-])c(N)n2)cc1-c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CFTR P13569 2/20 0.38
CYP2C9 P11712 1/20 0.38
GCGR P47871 3/20 0.32
AXL P30530 2/20 0.32
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
MEN1 O00255 1/20 0.31
MITF O75030 1/20 0.31
KMT2A Q03164 1/20 0.31
EIF4E P06730 1/20 0.31
AHR P35869 1/20 0.31
CXCR2 P25025 2/20 0.31
ALDH1A1 P00352 1/20 0.31
CNR1 P21554 1/20 0.30
MERTK Q12866 1/20 0.30
BRD4 O60885 1/20 0.30
ABL1 P00519 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2906883 1.00 CFTR (0.38) CFTRCYP2C9GCGRAXLGSK3A
SCHEMBL2907828 0.91 HPGD (0.36) GSK3AGSK3BSMN1; SMN2KMT2AALDH1A1
SCHEMBL2912050 0.91 HPGD (0.36) GSK3AGSK3BSMN1; SMN2KMT2AALDH1A1
SCHEMBL2910052 0.91 MAPT (0.34) CFTRAXLGSK3AGSK3BSMN1; SMN2
SCHEMBL2910524 0.91 MAPT (0.34) CFTRAXLGSK3AGSK3BSMN1; SMN2
SCHEMBL2908179 0.90 MET (0.34) AXLGSK3AGSK3BSMN1; SMN2MEN1
SCHEMBL2938731 0.90 MET (0.34) AXLGSK3AGSK3BSMN1; SMN2MEN1
SCHEMBL2913577 0.89 AHR (0.37) GCGRAXLGSK3AGSK3BSMN1; SMN2
SCHEMBL2911914 0.89 AHR (0.37) GCGRAXLGSK3AGSK3BSMN1; SMN2
SCHEMBL2911391 0.89 GSK3B (0.33) GSK3AGSK3BSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-B1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 NOVARTIS VACCINES & DIAGNOSTIC (US) 2010-08-11 EP disclosed