SCHEMBL29115477

SCHEMBL29115477

CNC(=O)c1ccc(N2CCNCC2)cc1Cl

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 5/20 0.56
USP28 Q96RU2 1/20 0.50
MAPK8 P45983 1/20 0.50
MAPK9 P45984 1/20 0.50
MAPK10 P53779 1/20 0.50
P2RX7 Q99572 1/20 0.48
HTR3E A5X5Y0 2/20 0.48
HTR3B O95264 2/20 0.48
HTR3A P46098 2/20 0.48
HTR3D Q70Z44 2/20 0.48
HTR3C Q8WXA8 2/20 0.48
SIGMAR1 Q99720 2/20 0.48
HTT P42858 2/20 0.48
TP53 P04637 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
HTR1A P08908 1/20 0.48
CYP2D6 P10635 1/20 0.48
THRB P10828 1/20 0.48
CYP2C9 P11712 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7653332 0.84 ADRB1 (0.58) ADRB1USP28P2RX7HTR3EHTR3B
SCHEMBL6868721 0.84 RAB9A (0.63) HTTHTR6PARP1TNK1RAB9A
SCHEMBL22625900 0.84 PARP1 (0.43) ADRB1USP28MAPK8MAPK9MAPK10
SCHEMBL4939443 0.84 ADRB1 (0.61) ADRB1USP28P2RX7HTR3EHTR3B
SCHEMBL25093446 0.83 PARP1 (0.48) ADRB1MAPK8MAPK9MAPK10HTR3E
SCHEMBL29960481 0.83 PARP1 (0.48) ADRB1MAPK8MAPK9MAPK10HTR3E
SCHEMBL14080465 0.82 ADRB1 (0.63) ADRB1USP28P2RX7HTR3EHTR3B
Hydrochloric Acid SCHEMBL29152389 0.82 PARP1 (0.48) ADRB1MAPK8MAPK9MAPK10HTR6
Hydrochloric Acid SCHEMBL15929282 0.81 ADRB1 (0.61) ADRB1USP28P2RX7HTR3EHTR3B
SCHEMBL29115571 0.81 ADRB1 (0.53) ADRB1USP28MAPK8MAPK9MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116710433-A Selective PARP1 inhibitor and application thereof 成都百裕制药股份有限公司 2023-09-05 CN disclosed
WO-2022222966-A1 SELECTIVE PARP1 INHIBITOR AND APPLICATION THEREOF 成都百裕制药股份有限公司 2022-10-27 WO disclosed