SCHEMBL29115488

SCHEMBL29115488

CN(C)CCNC(=O)c1ccc(N2CCNCC2)cc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
IKBKB O14920 1/20 0.44
ACKR3 P25106 1/20 0.44
USP25 Q9UHP3 3/20 0.44
USP28 Q96RU2 2/20 0.44
P2RX7 Q99572 1/20 0.42
ACVR1 Q04771 2/20 0.41
CYP1A2 P05177 1/20 0.41
RAD52 P43351 1/20 0.41
PRKD1 Q15139 1/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CDK2 P24941 2/20 0.41
BMPR1B O00238 1/20 0.40
BMPR1A P36894 1/20 0.40
TGFBR1 P36897 1/20 0.40
ACVRL1 P37023 1/20 0.40
CDK1 P06493 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29115473 0.86 P2RX7 (0.45) USP25USP28P2RX7ACVR1BMPR1B
SCHEMBL29115562 0.85 USP25 (0.44) USP25USP28P2RX7ACVR1CYP1A2
Hydrochloric Acid SCHEMBL708308 0.83 PARP1 (0.49) USP25USP28P2RX7ACVR1ALDH1A1
SCHEMBL20521486 0.83 ALDH1A1 (0.44) HTTSMN1; SMN2IKBKBACKR3USP25
SCHEMBL25093446 0.80 PARP1 (0.48) HTTIKBKBACVR1CYP1A2ALDH1A1
SCHEMBL29960481 0.80 PARP1 (0.48) HTTIKBKBACVR1CYP1A2ALDH1A1
Hydrochloric Acid SCHEMBL29152389 0.79 PARP1 (0.48) IKBKBACVR1BMPR1BBMPR1ATGFBR1
SCHEMBL29960471 0.77 ACVR1 (0.45) HTTUSP25USP28P2RX7ACVR1
SCHEMBL29115509 0.77 ACVR1 (0.60) HTTACVR1CYP1A2ALDH1A1HSD17B10
SCHEMBL5563304 0.76 ALDH1A1 (0.46) HTTSMN1; SMN2CYP1A2RAD52ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116710433-A Selective PARP1 inhibitor and application thereof 成都百裕制药股份有限公司 2023-09-05 CN disclosed
WO-2022222966-A1 SELECTIVE PARP1 INHIBITOR AND APPLICATION THEREOF 成都百裕制药股份有限公司 2022-10-27 WO disclosed