SCHEMBL29120406

SCHEMBL29120406

O=S(=O)(c1cccc2cnccc12)N1CCN(C(c2ccc(F)cc2)c2ccc(F)cc2)CC1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKD3 O94806 3/20 0.60
PRKCG P05129 3/20 0.60
PRKCB P05771 3/20 0.60
CYP3A4 P08684 3/20 0.60
PRKCA P17252 3/20 0.60
PRKCH P24723 3/20 0.60
PRKCI P41743 3/20 0.60
PRKCE Q02156 3/20 0.60
PRKCQ Q04759 3/20 0.60
PRKCZ Q05513 3/20 0.60
PRKCD Q05655 3/20 0.60
PRKD1 Q15139 3/20 0.60
ADORA3 P0DMS8 2/20 0.60
PRKACA P17612 2/20 0.60
PRKACG P22612 2/20 0.60
PRKACB P22694 2/20 0.60
KDM4E B2RXH2 1/20 0.60
CYP1A2 P05177 1/20 0.60
CYP2C19 P33261 1/20 0.60
ROCK2 O75116 13/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30423021 1.00 PRKD3 (0.60) PRKD3PRKCGPRKCBCYP3A4PRKCA
SCHEMBL13497829 0.82 ROCK2 (0.68) PRKD3PRKCGPRKCBCYP3A4PRKCA
SCHEMBL29770053 0.80 ROCK2 (0.77) PRKD3PRKCGPRKCBCYP3A4PRKCA
SCHEMBL7029110 0.79 PRKD3 (0.57) PRKD3PRKCGPRKCBCYP3A4PRKCA
SCHEMBL7315948 0.79 PRKD3 (0.74) PRKD3PRKCGPRKCBCYP3A4PRKCA
SCHEMBL10988523 0.78 ROCK2 (0.79) PRKD3PRKCGPRKCBCYP3A4PRKCA
SCHEMBL13497835 0.78 ROCK2 (0.64) PRKD3PRKCGPRKCBCYP3A4PRKCA
SCHEMBL2902584 0.78 CYP3A4 (0.72) PRKD3PRKCGPRKCBCYP3A4PRKCA
SCHEMBL6916059 0.77 ROCK2 (0.77) PRKD3PRKCGPRKCBCYP3A4PRKCA
SCHEMBL10985139 0.77 ROCK2 (0.77) PRKD3PRKCGPRKCBCYP3A4PRKCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116375685-B Fasudil derivative and preparation method and application thereof 沈阳药科大学 2023-12-12 CN disclosed
CN-116375685-A Fasudil derivative and preparation method and application thereof 沈阳药科大学 2023-07-04 CN disclosed