SCHEMBL29122807

SCHEMBL29122807

Nn1ncc2cc(Br)ccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.41
HDAC8 Q9BY41 1/20 0.39
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
ROCK1 Q13464 1/20 0.37
BACE1 P56817 2/20 0.37
NOS1 P29475 2/20 0.37
METAP2 P50579 2/20 0.37
CSNK2A1 P68400 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
CYP2A6 P11509 1/20 0.35
MCL1 Q07820 1/20 0.35
CHEK1 O14757 1/20 0.34
AURKA O14965 1/20 0.34
DAPK3 O43293 1/20 0.34
CSNK1A1 P48729 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27159441 0.84 KMO (0.51) KMOKDM4EMEN1ALDH1A1MAPT
SCHEMBL13137284 0.78 HDAC8 (0.40) KMOHDAC8KDM4EMEN1ALDH1A1
SCHEMBL3657596 0.76 CYP11B1 (0.47) KMOHDAC8KDM4EALDH1A1MAPT
SCHEMBL14765172 0.76 HDAC8 (0.39) KMOHDAC8KDM4EMEN1ALDH1A1
SCHEMBL11794 0.76 EGFR (0.46) KMOHDAC8ALDH1A1MAPTMCL1
SCHEMBL3660473 0.76 KMO (0.51) KMOHDAC8ALDH1A1MAPTKMT2A
SCHEMBL15798967 0.76 HDAC8 (0.39) KMOHDAC8KDM4EMEN1ALDH1A1
Hydrochloric Acid SCHEMBL11202185 0.74 HTR2A (0.44) KMOKDM4EMEN1ALDH1A1MAPT
SCHEMBL13468 0.74 HDAC8 (0.39) KMOHDAC8NOS1METAP2CSNK2A1
SCHEMBL25045382 0.72 HTR7 (0.39) HDAC8HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117120419-A KLK5 bicyclic heteroaromatic inhibitors 拜奥克里斯特制药公司 2023-11-24 CN disclosed