SCHEMBL30718282

SCHEMBL30718282

COc1cccc(-c2nc(Nc3ccccc3OC)nc3[nH]cc(Cl)c23)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.47
ALDH1A1 P00352 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
KDM4E B2RXH2 1/20 0.47
KMT2A Q03164 1/20 0.47
THRB P10828 1/20 0.43
ADORA2A P29274 2/20 0.43
ADORA1 P30542 2/20 0.43
GAA P10253 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
LRRK2 Q5S007 3/20 0.41
PIK3CG P48736 1/20 0.41
GSK3B P49841 1/20 0.41
CAMKK2 Q96RR4 1/20 0.41
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
TUBB4A P04350 1/20 0.40
TUBB P07437 1/20 0.40
TUBA3C P0DPH7 1/20 0.40
TUBA1B P68363 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29126163 1.00 MAPT (0.47) MAPTALDH1A1SMN1; SMN2KDM4EKMT2A
SCHEMBL29126151 0.78 HSP90AA1 (0.40) MAPTALDH1A1SMN1; SMN2KDM4EKMT2A
SCHEMBL29126098 0.76 LRRK2 (0.40) MAPTALDH1A1SMN1; SMN2KDM4EKMT2A
SCHEMBL30718280 0.73 MAPT (0.39) MAPTALDH1A1SMN1; SMN2KDM4EKMT2A
SCHEMBL27116596 0.71 PIK3CG (0.61) KMT2APIK3CGGSK3BCAMKK2EGFR
SCHEMBL30718279 0.71 LRRK2 (0.75) LRRK2IGF1R
SCHEMBL11813903 0.67 MAPT (0.83) MAPTALDH1A1SMN1; SMN2KDM4EKMT2A
SCHEMBL4544833 0.67 KCNH3 (0.59) MAPTALDH1A1SMN1; SMN2KDM4EKMT2A
SCHEMBL6237782 0.66 MAPT (0.93) MAPTALDH1A1SMN1; SMN2KDM4EKMT2A
SCHEMBL29609022 0.66 MAPT (0.93) MAPTALDH1A1SMN1; SMN2KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117247387-A Aromatic heterocyclic compound and preparation method thereof 上海翊石医药科技有限公司 2023-12-19 CN disclosed