SCHEMBL29129362

SCHEMBL29129362

COC(=O)c1nc(NC(=O)OC(C)(C)C)sc1C1CCOCC1

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LCK P06239 12/20 0.40
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
PIK3CG P48736 1/20 0.35
BRAF P15056 1/20 0.35
PI4KB Q9UBF8 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29129299 0.94 LCK (0.40) LCKCA1CA2PIK3CGBRAF
SCHEMBL25434541 0.81 RAF1 (0.35) LCKCA1CA2PIK3CGBRAF
SCHEMBL15348877 0.76 NPC1 (0.47) LCKCA1CA2PI4KBGAA
SCHEMBL29129275 0.76 NPSR1 (0.39) PIK3CG
SCHEMBL28733811 0.75 CA1 (0.44) LCKCA1CA2PI4KB
SCHEMBL1742407 0.75 LCK (0.46) LCKCA1CA2PI4KB
SCHEMBL29129336 0.75 ALDH1A1 (0.45) GAA
SCHEMBL23214462 0.75 LCK (0.46) LCKCA1CA2PI4KB
SCHEMBL23413609 0.75 CA1 (0.44) LCKCA1CA2PI4KB
SCHEMBL25147024 0.74 CNR2 (0.40) LCKPIK3CGGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117279896-A Amino substituted pyrido ring compounds, preparation method and application thereof 劲方医药科技(上海)有限公司 2023-12-22 CN disclosed
WO-2022214044-A1 AMINE-SUBSTITUTED PYRIDINE FUSED RING COMPOUNDS, PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2022-10-13 WO disclosed