SCHEMBL29129826

SCHEMBL29129826

O=C(Nc1ccc(Cl)cc1C(=O)c1ccccc1)c1ccncc1

nearest known ligand 0.84

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.74
SERPINE1 P05121 4/20 0.70
ALDH1A1 P00352 2/20 0.68
LMNA P02545 1/20 0.68
TP53 P04637 2/20 0.65
CYP1A2 P05177 1/20 0.62
CYP3A4 P08684 1/20 0.62
CYP2C9 P11712 1/20 0.62
CYP2C19 P33261 1/20 0.62
GAA P10253 1/20 0.60
KCNMA1 Q12791 2/20 0.59
SMN1; SMN2 Q16637 2/20 0.57
AKR1C4 P17516 1/20 0.55
AKR1C3 P42330 1/20 0.55
AKR1C2 P52895 1/20 0.55
AKR1C1 Q04828 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30694320 1.00 MAPT (0.74) MAPTSERPINE1ALDH1A1LMNATP53
SCHEMBL11571840 0.92 MAPT (0.86) MAPTSERPINE1ALDH1A1LMNATP53
SCHEMBL10413044 0.84 RAB9A (0.67) MAPTSERPINE1ALDH1A1LMNATP53
SCHEMBL31482309 0.83 POLB (0.71) MAPTALDH1A1TP53
SCHEMBL19860936 0.83 CCR9 (0.54) MAPTSERPINE1ALDH1A1LMNATP53
SCHEMBL420616 0.82 SERPINE1 (1.00) MAPTSERPINE1ALDH1A1LMNATP53
SCHEMBL6351321 0.82 SERPINE1 (0.89) MAPTSERPINE1KCNMA1AKR1C4AKR1C3
SCHEMBL15906641 0.82 CCR9 (0.64) MAPTALDH1A1LMNAGAAKCNMA1
SCHEMBL27611956 0.80 MAPT (0.72) MAPTSERPINE1ALDH1A1LMNATP53
SCHEMBL31384417 0.80 MAPT (0.67) MAPTSERPINE1ALDH1A1LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117285401-A Synthesis method of chiral N- (4-chloro-2- (hydroxy (phenyl) methyl) phenyl) isonicotinamide 中国科学院大连化学物理研究所 2023-12-26 CN claimed
CN-117285401-A Synthesis method of chiral N- (4-chloro-2- (hydroxy (phenyl) methyl) phenyl) isonicotinamide 中国科学院大连化学物理研究所 2023-12-26 CN disclosed
CN-117285401-A Synthesis method of chiral N- (4-chloro-2- (hydroxy (phenyl) methyl) phenyl) isonicotinamide 中国科学院大连化学物理研究所 2023-12-26 CN disclosed