SCHEMBL2912992

SCHEMBL2912992

O=C(NC1CCCCC1)C(C1CCCCC1)C1(Cc2ccc(F)cc2F)Nc2ccc(F)cc2N1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.45
RAB9A P51151 8/20 0.45
POLB P06746 1/20 0.45
ALDH1A1 P00352 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
LMNA P02545 1/20 0.38
IDO1 P14902 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
MLLT1 Q03111 1/20 0.36
EPHX1 P07099 1/20 0.36
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
GAA P10253 1/20 0.35
HTR2B P41595 1/20 0.35
ACKR3 P25106 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2909849 0.95 NPC1 (0.46) NPC1RAB9APOLBALDH1A1SMN1; SMN2
SCHEMBL3649621 0.84 NPC1 (0.40) NPC1RAB9APOLBSMN1; SMN2IDO1
SCHEMBL2912514 0.83 TP53 (0.40) NPC1RAB9APOLBSMN1; SMN2LMNA
SCHEMBL2912392 0.82 EPHX2 (0.48) NPC1RAB9ALMNASIGMAR1EPHX1
SCHEMBL3649148 0.81 NPC1 (0.42) NPC1RAB9APOLBALDH1A1SMN1; SMN2
SCHEMBL2914348 0.81 LMNA (0.44) NPC1RAB9AALDH1A1SMN1; SMN2LMNA
SCHEMBL2914853 0.81 MEN1 (0.46) NPC1RAB9APOLBLMNAEPHX1
SCHEMBL2907059 0.80 C3AR1 (0.39) NPC1RAB9APOLBALDH1A1SMN1; SMN2
SCHEMBL2907076 0.80 LMNA (0.47) NPC1RAB9APOLBALDH1A1SMN1; SMN2
SCHEMBL3651382 0.79 CNR2 (0.38) NPC1RAB9APOLBALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222645-A2 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS FXR AGONISTS F. Hoffmann-La Roche AG (CH) 2010-09-01 EP claimed
WO-2009062874-A2 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS FXR AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-05-22 WO claimed
EP-2222645-A2 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS FXR AGONISTS F. Hoffmann-La Roche AG (CH) 2010-09-01 EP disclosed
WO-2009062874-A2 BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS FXR AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-05-22 WO disclosed