SCHEMBL2913060

SCHEMBL2913060

O=[N+]([O-])N1CCCOc2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.44
PDK1 Q15118 1/20 0.43
ITGB2 P05107 1/20 0.42
ICAM1 P05362 1/20 0.42
ITGAL P20701 1/20 0.42
KMT2A Q03164 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
NPC1 O15118 1/20 0.39
POLB P06746 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
LMNA P02545 2/20 0.38
CRHBP P24387 2/20 0.38
CRHR2 Q13324 2/20 0.38
HTT P42858 1/20 0.38
TSHR P16473 2/20 0.38
CTSB P07858 2/20 0.37
GAA P10253 1/20 0.37
AR P10275 1/20 0.36
GRM7 Q14831 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12472476 0.75 PKM (0.37) KMT2APOLBLMNAGAAL3MBTL1
SCHEMBL301140 0.72 SMN1; SMN2 (0.50) NOTUMKMT2ASMN1; SMN2L3MBTL1
SCHEMBL9228795 0.72 NOTUM (0.49) NOTUMPDK1ITGB2ICAM1ITGAL
SCHEMBL5636846 0.72 ITGB2 (0.48) NOTUMPDK1ITGB2ICAM1ITGAL
SCHEMBL7345437 0.71 POLB (0.58) NOTUMKMT2APOLBSMN1; SMN2LMNA
SCHEMBL29877196 0.71 NOTUM (0.45) NOTUMPDK1ITGB2ICAM1ITGAL
SCHEMBL5636855 0.71 NOTUM (0.45) NOTUMPDK1ITGB2ICAM1ITGAL
SCHEMBL21455717 0.71 NOTUM (0.45) NOTUMPDK1ITGB2ICAM1ITGAL
Hydrochloric Acid SCHEMBL11437417 0.70 ITGB2 (0.46) NOTUMPDK1ITGB2ICAM1ITGAL
SCHEMBL19859267 0.69 NOTUM (0.58) NOTUMPDK1KMT2AHDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222647-A1 FUSED BICYCLIC DERIVATIVES OF 2,4-DIAMINOPYRIMIDINE AS ALK AND C-MET INHIBITORS Cephalon, Inc. (US) 2010-09-01 EP disclosed
WO-2008051547-A1 FUSED BICYCLIC DERIVATIVES OF 2,4-DIAMINOPYRIMIDINE AS ALK AND C-MET INHIBITORS CEPHALON, INC. (US) 2008-05-02 WO disclosed