SCHEMBL5636855

SCHEMBL5636855

O=NN1CCCOc2ccccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.45
PDK1 Q15118 1/20 0.44
ITGB2 P05107 1/20 0.43
ICAM1 P05362 1/20 0.43
ITGAL P20701 1/20 0.43
KMT2A Q03164 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
ALDH1A1 P00352 2/20 0.41
LMNA P02545 2/20 0.39
CRHBP P24387 2/20 0.39
CRHR2 Q13324 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
HTT P42858 1/20 0.39
POLB P06746 1/20 0.39
TSHR P16473 4/20 0.39
GRM7 Q14831 1/20 0.37
NPC1 O15118 1/20 0.37
AGTR2 P50052 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2362220 0.89 NOTUM (0.51) NOTUMPDK1ITGB2ICAM1ITGAL
SCHEMBL30395562 0.89 NOTUM (0.51) NOTUMPDK1ITGB2ICAM1ITGAL
SCHEMBL11431097 0.79 ALDH1A1 (0.59) KMT2AALDH1A1LMNASMN1; SMN2HTT
SCHEMBL11436384 0.74 HTR2A (0.42) NOTUMPDK1ITGB2ICAM1ITGAL
SCHEMBL9228795 0.73 NOTUM (0.49) NOTUMPDK1ITGB2ICAM1ITGAL
SCHEMBL5636846 0.73 ITGB2 (0.48) NOTUMPDK1ITGB2ICAM1ITGAL
SCHEMBL18650412 0.72 ALDH1A1 (0.40) NOTUMKMT2AALDH1A1SMN1; SMN2TSHR
SCHEMBL29877196 0.72 NOTUM (0.45) NOTUMPDK1ITGB2ICAM1ITGAL
Hydrochloric Acid SCHEMBL11437417 0.71 ITGB2 (0.46) NOTUMPDK1ITGB2ICAM1ITGAL
SCHEMBL2913060 0.71 NOTUM (0.44) NOTUMPDK1ITGB2ICAM1ITGAL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39679-E1 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2007-06-05 US disclosed
US-6713471-B1 SUCH AS TERT-BUTYL-1-METHYL-6,7,9,12-TETRAHYDRO-5H-PYRIDO-(4,3-B)(1,4) THIAZEPINO(2,3,4-HI)INDOLE-11(10H)-CARBOXYLATE; SEROTONIN AGONISTS AND ANTAGONISTS; CENTRAL NERVOUS SYSTEM DISORDERS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-03-30 US disclosed