SCHEMBL2913172

SCHEMBL2913172

CC1CCCCC1(C(N)=O)c1ccccc1C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.48
TAS1R3 Q7RTX0 2/20 0.36
TAS1R1 Q7RTX1 2/20 0.36
TAS1R2 Q8TE23 2/20 0.36
PDE4D Q08499 1/20 0.36
GAA P10253 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
BACE1 P56817 1/20 0.35
KCNH2 Q12809 1/20 0.35
EPHX2 P34913 1/20 0.35
PDE7A Q13946 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6472112 0.84 HDAC4 (0.45) HDAC4PDE4DGAAKDM4EALDH1A1
SCHEMBL18742726 0.73 HDAC4 (0.63) HDAC4GAAHDAC3HDAC1HDAC2
SCHEMBL29661878 0.71 HDAC4 (0.60) HDAC4GAAHDAC3HDAC1HDAC2
SCHEMBL5342025 0.71 HDAC4 (0.60) HDAC4GAAHDAC3HDAC1HDAC2
SCHEMBL14232917 0.70 HDAC4 (0.46) HDAC4GAA
SCHEMBL2435589 0.70 KDM4E (0.43) KDM4EALDH1A1
SCHEMBL6597123 0.69 SLC6A2 (0.41) ALDH1A1
SCHEMBL2913178 0.69 GAA (0.44) HDAC4GAATDP1KDM4EALDH1A1
SCHEMBL9330906 0.68 AKR1C1 (0.50) HDAC4
SCHEMBL9386533 0.68 RXRA (0.36) HDAC4GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2214487-A1 NOVEL SEH INHIBITORS AND THEIR USE GlaxoSmithKline LLC (US) 2010-08-11 EP disclosed
WO-2009049157-A1 NOVEL SEH INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-04-16 WO disclosed