SCHEMBL29132274

SCHEMBL29132274

CC(C)(C)OC(=O)N1CCC(Cc2ccc(CC3CCN(c4cc(B5OC(C)(C)C(C)(C)O5)ccn4)CC3)cc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 12/20 0.48
USP30 Q70CQ3 2/20 0.47
FAAH O00519 1/20 0.42
HRH3 Q9Y5N1 1/20 0.39
WNT3A P56704 1/20 0.38
GNRHR P30968 1/20 0.38
HDAC1 Q13547 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29132290 0.88 GPR119 (0.46) GPR119USP30FAAHHRH3
SCHEMBL1073012 0.86 USP30 (0.48) GPR119USP30WNT3A
SCHEMBL29504310 0.86 USP30 (0.48) GPR119USP30WNT3A
SCHEMBL29132112 0.85 GPR119 (0.48) GPR119USP30HRH3
SCHEMBL3375291 0.85 USP30 (0.53) GPR119USP30FAAHGNRHR
SCHEMBL29039949 0.82 USP30 (0.51) GPR119USP30FAAHHDAC1
SCHEMBL1363539 0.82 USP30 (0.48) GPR119USP30GNRHR
SCHEMBL29132200 0.82 GPR119 (0.54) GPR119USP30FAAHHDAC1
SCHEMBL25420114 0.80 USP30 (0.51) GPR119USP30FAAHGNRHR
SCHEMBL26187097 0.80 USP30 (0.56) GPR119USP30FAAHGNRHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4308557-A1 INDAZOLE BASED COMPOUNDS AND ASSOCIATED METHODS OF USE Arvinas Operations, Inc. (US) 2024-01-24 EP disclosed
CN-117321046-A Indazole-based compounds and related methods of use 阿维纳斯企业公司 2023-12-29 CN disclosed
WO-2022198112-A1 INDAZOLE BASED COMPOUNDS AND ASSOCIATED METHODS OF USE ARVINAS OPERATIONS, INC. (US) 2022-09-22 WO disclosed