SCHEMBL29132280

SCHEMBL29132280

CC(C)(C)OC(=O)N1CCN(CC2CCN(c3cc(Br)ccn3)CC2)CC1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 10/20 0.52
FAAH O00519 1/20 0.43
CNR1 P21554 1/20 0.43
FPR2 P25090 2/20 0.42
LRRK2 Q5S007 1/20 0.42
HRH3 Q9Y5N1 2/20 0.41
CKS1B P61024 1/20 0.41
SKP1 P63208 1/20 0.41
SKP2 Q13309 1/20 0.41
FPR3 P25089 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30066214 0.96 GPR119 (0.52) GPR119FAAHCNR1FPR2LRRK2
SCHEMBL24671505 0.96 GPR119 (0.52) GPR119FAAHCNR1FPR2LRRK2
SCHEMBL30179976 0.86 GPR119 (0.54) GPR119LRRK2CKS1BSKP1SKP2
SCHEMBL901264 0.86 GPR119 (0.54) GPR119LRRK2CKS1BSKP1SKP2
SCHEMBL29132200 0.86 GPR119 (0.54) GPR119FAAH
SCHEMBL29132186 0.84 GPR119 (0.48) GPR119FAAHCNR1
SCHEMBL29132207 0.83 GPR119 (0.52) GPR119FAAH
SCHEMBL7650536 0.83 GPR119 (0.55) GPR119FAAHCNR1CKS1BSKP1
SCHEMBL29132048 0.82 GPR119 (0.57) GPR119
SCHEMBL31584217 0.82 GPR119 (0.50) GPR119FAAHCNR1LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4308557-A1 INDAZOLE BASED COMPOUNDS AND ASSOCIATED METHODS OF USE Arvinas Operations, Inc. (US) 2024-01-24 EP disclosed
CN-117321046-A Indazole-based compounds and related methods of use 阿维纳斯企业公司 2023-12-29 CN disclosed
WO-2022198112-A1 INDAZOLE BASED COMPOUNDS AND ASSOCIATED METHODS OF USE ARVINAS OPERATIONS, INC. (US) 2022-09-22 WO disclosed