SCHEMBL29133075

SCHEMBL29133075

COCc1cc(-c2cc(OC)cnn2)ccc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.38
CYP11B2 P19099 2/20 0.38
NR1I2 O75469 1/20 0.35
NR1I3 Q14994 1/20 0.35
MAPT P10636 2/20 0.34
TSHR P16473 1/20 0.34
NPY1R P25929 1/20 0.34
NPY2R P49146 1/20 0.34
NOTUM Q6P988 1/20 0.34
GUSB P08236 1/20 0.34
CASP1 P29466 1/20 0.33
TUBB4A P04350 1/20 0.33
TUBB P07437 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
TUBA1B P68363 1/20 0.33
TUBA4A P68366 1/20 0.33
TUBB4B P68371 1/20 0.33
TUBB3 Q13509 1/20 0.33
TUBB2A Q13885 1/20 0.33
TUBB8 Q3ZCM7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30622182 1.00 CYP11B1 (0.38) CYP11B1CYP11B2NR1I2NR1I3MAPT
SCHEMBL30622232 0.78 SLC6A2 (0.40) NR1I2NR1I3NOTUMP2RX7DHODH
SCHEMBL29133196 0.78 SLC6A2 (0.40) NR1I2NR1I3NOTUMP2RX7DHODH
SCHEMBL30622194 0.76 P2RX7 (0.52) NR1I2NR1I3MAPTNOTUMP2RX7
SCHEMBL5780833 0.76 CASP1 (0.44) CYP11B1CYP11B2MAPTCASP1GRIN1
SCHEMBL29133088 0.76 P2RX7 (0.52) NR1I2NR1I3MAPTNOTUMP2RX7
SCHEMBL26654427 0.73 P2RX7 (0.39) NR1I2NR1I3MAPTNOTUMP2RX7
SCHEMBL30622200 0.73 P2RX7 (0.39) NR1I2NR1I3MAPTNOTUMP2RX7
SCHEMBL24252449 0.72 SLC6A4 (0.46) CYP11B1CYP11B2MAPTTUBB4ATUBB
SCHEMBL29133194 0.72 CYP2D6 (0.44) CYP11B1CYP11B2P2RX7PIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117088884-A Imidazopyridazine derivatives as GABAA receptor modulators, pharmaceutical compositions and uses 上海赛默罗德生物科技有限公司 2023-11-21 CN disclosed