SCHEMBL29133097

SCHEMBL29133097

COCc1cc(-c2nnco2)ccc1Br

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.52
HPGD P15428 1/20 0.52
MAPK1 P28482 1/20 0.52
NOTUM Q6P988 10/20 0.52
TSHR P16473 1/20 0.49
RAB9A P51151 4/20 0.46
NPC1 O15118 3/20 0.46
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.43
TLR8 Q9NR97 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22325385 0.78 HPGD (0.57) ALDH1A1HPGDMAPK1NOTUMTSHR
SCHEMBL31488513 0.78 HPGD (0.57) ALDH1A1HPGDMAPK1NOTUMTSHR
SCHEMBL29133064 0.77 NOTUM (0.43) ALDH1A1HPGDMAPK1NOTUMTSHR
SCHEMBL29133160 0.77 SMN1; SMN2 (0.41) ALDH1A1HPGDMAPK1NOTUMRAB9A
SCHEMBL29133017 0.76 DGAT1 (0.50) ALDH1A1HPGDMAPK1NOTUMRAB9A
SCHEMBL1459174 0.75 TSHR (0.62) ALDH1A1HPGDMAPK1NOTUMTSHR
SCHEMBL30221689 0.75 TSHR (0.62) ALDH1A1HPGDMAPK1NOTUMTSHR
SCHEMBL30622248 0.75 KDM4E (0.49) ALDH1A1HPGDMAPK1NOTUMRAB9A
SCHEMBL792274 0.73 PTPN1 (0.36) ALDH1A1HPGDRAB9ANPC1KDM4E
SCHEMBL29133117 0.73 HDAC6 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117088884-A Imidazopyridazine derivatives as GABAA receptor modulators, pharmaceutical compositions and uses 上海赛默罗德生物科技有限公司 2023-11-21 CN disclosed