SCHEMBL29133064

SCHEMBL29133064

COCc1nnc(-c2ccc(Br)c(COC)c2)o1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 3/20 0.43
MAPT P10636 9/20 0.42
POLB P06746 5/20 0.42
KDM4E B2RXH2 4/20 0.42
HSD17B10 Q99714 4/20 0.42
LMNA P02545 3/20 0.42
ALDH1A1 P00352 3/20 0.42
MAPK1 P28482 3/20 0.42
HPGD P15428 3/20 0.42
TSHR P16473 3/20 0.42
USP2 O75604 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
HTT P42858 1/20 0.41
RXFP1 Q9HBX9 1/20 0.40
KMT2A Q03164 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TP53 P04637 1/20 0.39
QPCT Q16769 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30622193 0.88 TLR8 (0.43) NOTUMMAPTPOLBKDM4EHSD17B10
SCHEMBL29133160 0.86 SMN1; SMN2 (0.41) NOTUMMAPTPOLBKDM4EHSD17B10
SCHEMBL29133041 0.84 KDM4E (0.52) NOTUMMAPTPOLBKDM4EHSD17B10
SCHEMBL29133017 0.84 DGAT1 (0.50) NOTUMMAPTPOLBKDM4EHSD17B10
SCHEMBL30622248 0.83 KDM4E (0.49) NOTUMMAPTPOLBKDM4EHSD17B10
SCHEMBL29133007 0.82 MAPT (0.48) MAPTPOLBALDH1A1KMT2ARAB9A
SCHEMBL29133117 0.81 HDAC6 (0.45)
SCHEMBL5115763 0.80 MAPT (0.58) MAPTPOLBKDM4EHSD17B10LMNA
SCHEMBL29133055 0.80 ALDH1A1 (0.52) MAPTPOLBKDM4EALDH1A1MAPK1
SCHEMBL29133097 0.77 ALDH1A1 (0.52) NOTUMMAPTKDM4ELMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117088884-A Imidazopyridazine derivatives as GABAA receptor modulators, pharmaceutical compositions and uses 上海赛默罗德生物科技有限公司 2023-11-21 CN disclosed