SCHEMBL29133150

SCHEMBL29133150

COc1cc(-c2nnccc2C)ccc1Br

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 4/20 0.39
MAOB P27338 1/20 0.39
NQO2 P16083 1/20 0.38
GRM2 Q14416 1/20 0.37
ABCG2 Q9UNQ0 3/20 0.37
ABCB1 P08183 2/20 0.37
ABCC1 P33527 2/20 0.37
MAPT P10636 2/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
MAPK1 P28482 1/20 0.35
POLB P06746 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
DHFR P00374 1/20 0.34
GRM4 Q14833 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30622149 1.00 S1PR1 (0.39) S1PR1MAOBNQO2GRM2ABCG2
SCHEMBL30622206 0.88 MAOB (0.37) S1PR1MAOBGRM2ABCG2ABCB1
SCHEMBL29133015 0.88 MAOB (0.37) S1PR1MAOBGRM2ABCG2ABCB1
SCHEMBL4312617 0.74 ALDH1A1 (0.54) MAOBNQO2ABCG2ABCB1ABCC1
SCHEMBL29133201 0.74 MAPT (0.39) S1PR1MAOBABCG2ABCB1ABCC1
SCHEMBL30622169 0.74 MAPT (0.39) S1PR1MAOBABCG2ABCB1ABCC1
SCHEMBL24185298 0.73 TRPV1 (0.39) MAPTALDH1A1HPGDMAPK1
SCHEMBL28279253 0.72 DYRK1A (0.51) MAOBMAPTALDH1A1HPGD
SCHEMBL31300130 0.70 MAPT (0.49) S1PR1MAPTALDH1A1
SCHEMBL29133104 0.70 CLK1 (0.46) MAOBGRM2ALDH1A1HPGDMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117088884-A Imidazopyridazine derivatives as GABAA receptor modulators, pharmaceutical compositions and uses 上海赛默罗德生物科技有限公司 2023-11-21 CN disclosed