SCHEMBL29133201

SCHEMBL29133201

COc1cc(-c2cccnn2)ccc1Br

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.39
KDM4E B2RXH2 5/20 0.39
ALDH1A1 P00352 4/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
HPGD P15428 2/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
ACACA Q13085 1/20 0.38
ABCB1 P08183 1/20 0.38
ABCC1 P33527 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
NPC1 O15118 3/20 0.37
RAB9A P51151 3/20 0.37
GRM4 Q14833 1/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
MAPK1 P28482 2/20 0.37
HSD17B10 Q99714 2/20 0.37
USP2 O75604 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30622169 1.00 MAPT (0.39) MAPTKDM4EALDH1A1SMN1; SMN2HPGD
SCHEMBL27736352 0.85 ALDH1A1 (0.50) MAPTKDM4EALDH1A1SMN1; SMN2HPGD
SCHEMBL38660064 0.81 GAA (0.51) MAPTKDM4EALDH1A1SMN1; SMN2HPGD
SCHEMBL29141516 0.79 ERN1 (0.51) MAPTKDM4EALDH1A1SMN1; SMN2HPGD
SCHEMBL27982666 0.78 KMO (0.49) GRM4MEN1KMT2AL3MBTL1
SCHEMBL29133015 0.76 MAOB (0.37) MAPTKDM4EALDH1A1HPGDABCB1
SCHEMBL30622206 0.76 MAOB (0.37) MAPTKDM4EALDH1A1HPGDABCB1
SCHEMBL30622160 0.76 HDAC4 (0.42) KDM4EALDH1A1RAB9AMAPK1PRMT5
SCHEMBL28878342 0.76 HDAC4 (0.42) KDM4EALDH1A1RAB9AMAPK1PRMT5
SCHEMBL4312617 0.75 ALDH1A1 (0.54) MAPTALDH1A1HPGDABCB1ABCC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117088884-A Imidazopyridazine derivatives as GABAA receptor modulators, pharmaceutical compositions and uses 上海赛默罗德生物科技有限公司 2023-11-21 CN disclosed