SCHEMBL29133316

SCHEMBL29133316

COc1ccc(Cn2ncc(C)c2[Na])cc1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 12/20 0.52
MCHR1 Q99705 1/20 0.51
ALDH1A1 P00352 2/20 0.47
MAPT P10636 2/20 0.47
KDM4E B2RXH2 1/20 0.47
ALOX15 P16050 1/20 0.47
DCTPP1 Q9H773 1/20 0.46
LMNA P02545 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PDE1A P54750 2/20 0.44
PDE1B Q01064 2/20 0.44
PDE1C Q14123 2/20 0.44
UCHL1 P09936 1/20 0.44
CMA1 P23946 1/20 0.44
PKM P14618 1/20 0.43
PKLR P30613 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13964565 0.84 NPBWR1 (0.55) NPBWR1MCHR1ALDH1A1MAPTKDM4E
SCHEMBL25045656 0.83 NPBWR1 (0.57) NPBWR1MCHR1ALDH1A1MAPTKDM4E
SCHEMBL18096396 0.81 NPBWR1 (0.52) NPBWR1MCHR1ALDH1A1MAPTKDM4E
SCHEMBL1491119 0.81 TSHR (0.67) NPBWR1MCHR1ALDH1A1MAPTKDM4E
SCHEMBL25723425 0.79 NPBWR1 (0.64) NPBWR1MCHR1ALDH1A1SMN1; SMN2PDE1A
SCHEMBL25833185 0.78 NPBWR1 (0.49) NPBWR1MCHR1ALDH1A1MAPTKDM4E
SCHEMBL28496573 0.77 NPBWR1 (0.51) NPBWR1MCHR1ALDH1A1MAPTKDM4E
SCHEMBL16252260 0.77 UCHL1 (0.54) NPBWR1MCHR1ALDH1A1MAPTKDM4E
SCHEMBL4679664 0.77 NPBWR1 (0.61) NPBWR1MCHR1ALDH1A1SMN1; SMN2PDE1A
SCHEMBL25756148 0.77 NPBWR1 (0.61) NPBWR1MCHR1ALDH1A1SMN1; SMN2PDE1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117285547-A Macrocyclic compounds as modulators of CFTR, pharmaceutical compositions thereof, their use and methods of preparation 弗特克斯药品有限公司 2023-12-26 CN disclosed