SCHEMBL29134489

SCHEMBL29134489

CC(C)(C)OC(=O)N1CCc2cc(Br)ccc2C1C(F)F

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ABHD6 Q9BV23 3/20 0.42
GHSR Q92847 11/20 0.41
NR1H2 P55055 3/20 0.41
NR1H3 Q13133 1/20 0.41
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
USP30 Q70CQ3 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20504327 0.90 GHSR (0.44) ABHD6GHSRNR1H2NR1H3
SCHEMBL20504328 0.90 GHSR (0.44) ABHD6GHSRNR1H2NR1H3
SCHEMBL29676621 0.83 NR1H2 (0.43) ABHD6GHSRNR1H2NR1H3ESR1
SCHEMBL12280043 0.83 NR1H2 (0.43) ABHD6GHSRNR1H2NR1H3ESR1
SCHEMBL19026010 0.80 GHSR (0.44) GHSRNR1H2NR1H3
SCHEMBL33532880 0.80 UCHL1 (0.52) ABHD6GHSRNR1H2NR1H3USP30
SCHEMBL19026148 0.80 GHSR (0.44) GHSRNR1H2NR1H3
SCHEMBL19025987 0.80 GHSR (0.44) GHSRNR1H2NR1H3
SCHEMBL27276905 0.79 ESR1 (0.51) GHSRNR1H2NR1H3ESR1ESR2
SCHEMBL2792433 0.78 CYP2D6 (0.44) ABHD6NR1H2NR1H3ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4313967-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2024-02-07 EP disclosed
CN-117120429-A KHK inhibitor 吉利德科学公司 2023-11-24 CN disclosed
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed