SCHEMBL29134531

SCHEMBL29134531

COc1cc(Sc2cc(Br)ccc2OC)ccc1C#N

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 12/20 0.68
MAOB P27338 4/20 0.51
MAOA P21397 2/20 0.51
KDM4E B2RXH2 1/20 0.42
USP2 O75604 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TUBB4A P04350 1/20 0.40
TUBB P07437 1/20 0.40
TUBA3C P0DPH7 1/20 0.40
TUBA1B P68363 1/20 0.40
TUBA4A P68366 1/20 0.40
TUBB4B P68371 1/20 0.40
TUBB3 Q13509 1/20 0.40
TUBB2A Q13885 1/20 0.40
TUBB8 Q3ZCM7 1/20 0.40
TUBA3E Q6PEY2 1/20 0.40
TUBA1A Q71U36 1/20 0.40
TUBA1C Q9BQE3 1/20 0.40
TUBB6 Q9BUF5 1/20 0.40
TUBB2B Q9BVA1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29134827 0.88 AR (0.53) ARMAOBMAOAKDM4EUSP2
SCHEMBL29134917 0.83 MAOB (0.56) ARMAOBMAOAALDH1A1TUBB4A
SCHEMBL29134515 0.82 AR (0.64) ARMAOBMAOAIMPDH2PGR
SCHEMBL286644 0.80 AR (0.53) ARKDM4EUSP2ALDH1A1IDH1
SCHEMBL29964800 0.77 ALDH1A1 (0.61) ARMAOBMAOAKDM4EUSP2
SCHEMBL393816 0.77 ALDH1A1 (0.61) ARMAOBMAOAKDM4EUSP2
SCHEMBL31345528 0.76 ALDH1A1 (0.56) ARKDM4EALDH1A1TUBB4ATUBB
SCHEMBL5094814 0.76 AR (0.62) ARMAOBMAOAKDM4EUSP2
SCHEMBL20389510 0.74 MAOB (0.66) ARMAOBMAOAKDM4EALDH1A1
SCHEMBL31061245 0.71 AR (1.00) ARMAOBMAOAIMPDH2IMPDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117120429-A KHK inhibitor 吉利德科学公司 2023-11-24 CN disclosed