SCHEMBL29134978

SCHEMBL29134978

Fc1ccc(-c2cccc(C(F)(F)F)c2)cn1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 4/20 0.55
GRIN2B Q13224 4/20 0.55
DYRK1A Q13627 1/20 0.54
DYRK2 Q92630 1/20 0.54
ALDH1A1 P00352 2/20 0.50
SCN2A Q99250 2/20 0.50
GAA P10253 1/20 0.50
ATM Q13315 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.48
IDO1 P14902 1/20 0.47
PARP1 P09874 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
NR3C1 P04150 1/20 0.47
PGR P06401 1/20 0.47
MAOB P27338 2/20 0.46
HRH1 P35367 1/20 0.46
HRH4 Q9H3N8 1/20 0.46
KDM1A O60341 1/20 0.45
ADORA2A P29274 1/20 0.44
ADORA1 P30542 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15394358 0.85 KIF11 (0.53) GRIN1GRIN2BDYRK1ADYRK2ALDH1A1
SCHEMBL16068085 0.83 GRIN1 (0.55) GRIN1GRIN2BALDH1A1SCN2AGAA
SCHEMBL8274248 0.81 GRIN1 (0.56) GRIN1GRIN2BALDH1A1SCN2AGAA
SCHEMBL11158643 0.81 CCNA2 (0.55) GRIN1GRIN2BDYRK1ADYRK2ALDH1A1
SCHEMBL30704262 0.81 MAP4K4 (0.62) ALDH1A1SCN2AGAAATML3MBTL1
SCHEMBL28051302 0.81 MAP4K4 (0.62) ALDH1A1SCN2AGAAATML3MBTL1
SCHEMBL13803129 0.81 ALDH1A1 (0.47) GRIN1GRIN2BDYRK1ADYRK2ALDH1A1
SCHEMBL29678302 0.79 TSHR (0.58) ALDH1A1SCN2AIDO1PGRMAOB
SCHEMBL1263144 0.79 TSHR (0.58) ALDH1A1SCN2AIDO1PGRMAOB
SCHEMBL6241092 0.78 CTSS (0.58) GRIN1GRIN2BALDH1A1SCN2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117343004-A Preparation method of 2-aminopyridine compound 易简和成(江苏)医药科技有限公司 2024-01-05 CN disclosed