SCHEMBL29135632

SCHEMBL29135632

CC(C)(C)OC(=O)NCCCOc1ccc(F)cc1COS(C)(=O)=O

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA1 P00915 8/20 0.47
CA2 P00918 8/20 0.47
CA12 O43570 5/20 0.47
CA9 Q16790 5/20 0.47
AXL P30530 2/20 0.47
SCN9A Q15858 1/20 0.41
BRD4 O60885 1/20 0.39
NQO2 P16083 1/20 0.39
DRD2 P14416 4/20 0.39
CYP1A1 P04798 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2B6 P20813 1/20 0.39
CYP2C19 P33261 1/20 0.39
CYP3A43 Q9HB55 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21513609 0.84 CA12 (0.49) CA1CA2CA12CA9AXL
SCHEMBL29135647 0.83 SSTR4 (0.41)
SCHEMBL23020273 0.83 CA12 (0.46) CA1CA2CA12CA9AXL
SCHEMBL29293585 0.82 SCN9A (0.48) CA1CA2CA12CA9AXL
SCHEMBL29135644 0.80 MKNK2 (0.44) NQO2
SCHEMBL30786834 0.80 AAK1 (0.44)
SCHEMBL29135633 0.80 AAK1 (0.44)
SCHEMBL29135641 0.80 MKNK2 (0.44) NQO2
SCHEMBL28963091 0.80 SCN9A (0.47) CA1CA2CA12CA9AXL
SCHEMBL16946788 0.79 SCN9A (0.46) CA1CA2CA12CA9AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117229295-A Nitrogen-containing macrocyclic compound, and preparation method and medical application thereof 中国医药研究开发中心有限公司 2023-12-15 CN disclosed