SCHEMBL29137722

SCHEMBL29137722

COc1nccc2ccc(Nc3ccc(C(C)Nc4ncc(CC(=O)OC(C)(C)C)cn4)cc3)nc12

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRAF P15056 10/20 0.39
VNN1 O95497 1/20 0.34
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
NPR3 P17342 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C8 P10632 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
PLK1 P53350 2/20 0.32
FLT4 P35916 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA2B P29275 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29137721 0.89 CAMK2D (0.40) BRAFVNN1HDAC3HDAC1HDAC2
SCHEMBL29137741 0.82 EZH2 (0.38) BRAFVNN1HDAC3HDAC1HDAC2
SCHEMBL29137743 0.82 EZH2 (0.39) BRAFVNN1HDAC3HDAC1HDAC2
SCHEMBL30768169 0.80 NPC1 (0.41) BRAFCYP1A2CYP3A4CYP2C19PLK1
SCHEMBL23169690 0.77 PCSK9 (0.31)
SCHEMBL32661517 0.77 AURKA (0.34) BRAF
SCHEMBL32662613 0.74 BRD4 (0.42) HDAC1
SCHEMBL31563705 0.74 BRD4 (0.42) HDAC1
SCHEMBL23169315 0.73 EZH2 (0.50) ADORA2AADORA2B
SCHEMBL32661546 0.72 ACACB (0.37) BRAFVNN1HDAC3HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117384153-A Methyltransferase inhibitors and uses thereof 上海赛岚生物科技有限公司 2024-01-12 CN disclosed