SCHEMBL29138030

SCHEMBL29138030

COc1cc2c(cc1S(N)(=O)=O)C(=O)COC2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 4/20 0.49
CYP3A4 P08684 1/20 0.44
CA2 P00918 5/20 0.40
CA1 P00915 4/20 0.40
CA12 O43570 4/20 0.40
CA9 Q16790 4/20 0.40
TSHR P16473 1/20 0.38
BRD4 O60885 1/20 0.37
CA7 P43166 1/20 0.37
ACHE P22303 1/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 2/20 0.36
MAPK1 P28482 2/20 0.36
RAB9A P51151 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
NPC1 O15118 1/20 0.36
XBP1 P17861 1/20 0.36
PAX8 Q06710 1/20 0.36
ATM Q13315 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30688577 0.84 CYP3A4 (0.61) CYP3A4CA2CA1CA9CA7
SCHEMBL30688578 0.84 CYP3A4 (0.61) CYP3A4CA2CA1CA9CA7
SCHEMBL27117787 0.83 CYP3A4 (0.47) PKMCYP3A4TSHRACHEALDH1A1
SCHEMBL30759602 0.83 CYP3A4 (0.47) PKMCYP3A4TSHRACHEALDH1A1
SCHEMBL31217500 0.77 CYP3A4 (0.42) CYP3A4ALDH1A1MAPTGAA
SCHEMBL29138028 0.77 CYP3A4 (0.42) CYP3A4ALDH1A1MAPTGAA
SCHEMBL31525908 0.74 PKM (0.58) PKMCA2CA1CA12CA9
SCHEMBL10640095 0.74 PKM (0.58) PKMCA2CA1CA12CA9
SCHEMBL31172537 0.72 PKM (0.56) PKMCYP3A4CA2CA1CA12
SCHEMBL11688578 0.72 PKM (0.70) PKMCA2CA1CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117343036-A Isochroman compound, and pharmaceutical composition and application thereof 江苏联环药业股份有限公司 2024-01-05 CN disclosed