SCHEMBL29138028

SCHEMBL29138028

COc1cc2c(cc1C(N)=O)C(=O)COC2

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.42
IRAK4 Q9NWZ3 6/20 0.37
MKNK1 Q9BUB5 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36
PARP1 P09874 1/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
KMT2A Q03164 1/20 0.36
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
CHEK1 O14757 1/20 0.35
GLA P06280 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
PARP15 Q460N3 1/20 0.34
PARP10 Q53GL7 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34
ADORA1 P30542 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31217500 1.00 CYP3A4 (0.42) CYP3A4IRAK4MKNK1MKNK2PARP1
SCHEMBL30688578 0.81 CYP3A4 (0.61) CYP3A4KDM4EALDH1A1KMT2AMAPT
SCHEMBL30688577 0.81 CYP3A4 (0.61) CYP3A4KDM4EALDH1A1KMT2AMAPT
SCHEMBL3968873 0.81 TUBB4A (0.42) IRAK4KDM4EALDH1A1KMT2ACHEK1
SCHEMBL27117787 0.77 CYP3A4 (0.47) CYP3A4KDM4EALDH1A1MAPTHTT
SCHEMBL30759602 0.77 CYP3A4 (0.47) CYP3A4KDM4EALDH1A1MAPTHTT
SCHEMBL29138030 0.77 PKM (0.49) CYP3A4ALDH1A1MAPTGAA
SCHEMBL12515332 0.70 CYP3A4 (0.52) CYP3A4MKNK1MKNK2KDM4EALDH1A1
SCHEMBL3967663 0.69 CYP1A2 (0.41) CYP3A4KDM4EALDH1A1MAPTCHEK1
SCHEMBL3967662 0.69 CYP1A2 (0.41) CYP3A4KDM4EALDH1A1MAPTCHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117343036-A Isochroman compound, and pharmaceutical composition and application thereof 江苏联环药业股份有限公司 2024-01-05 CN claimed
CN-117343036-A Isochroman compound, and pharmaceutical composition and application thereof 江苏联环药业股份有限公司 2024-01-05 CN disclosed